• Retatrutide 2381089-83-2

  • Retatrutide 2381089-83-2

  • Retatrutide 2381089-83-2

Retatrutide 2381089-83-2

Retatrutide (CAS No. 2381089-83-2) is a groundbreaking, triple-receptor agonist peptide that targets key pathways in metabolic regulation. By combining the actions of GLP-1, GIP, and Glucagon receptors, Retatrutide offers a novel approach for treating obesity and type-2 diabetes, both of which are major challenges in today’s healthcare landscape.

Product Description

Key Features & Advantages

 

Triple-Action Mechanism of Action

 

Retatrutide's efficacy lies in its triple receptor activation:

 

● GLP-1 Agonist: Enhances glucose-dependent insulin secretion, promotes satiety, and slows gastric emptying.

 

● GIP Agonist: Regulates appetite control and insulin sensitivity, promoting overall metabolic balance.

 

● Glucagon Receptor Activation: Increases energy expenditure and fat oxidation, contributing to weight loss.

 

This integrated approach to metabolic regulation makes Retatrutide a promising candidate for treating obesity, metabolic syndrome, and type-2 diabetes with more comprehensive therapeutic effects compared to traditional single-target peptides.

 

Potent Weight Loss Effects

 

Retatrutide has shown substantial weight loss in clinical trials, making it a highly sought-after peptide for obesity management. Its dual effect on glucose metabolism and appetite suppression helps patients experience significant body fat reduction, improving both health outcomes and quality of life.

 

Improved Glycemic Control

 

As a dual-action peptide, Retatrutide enhances insulin secretion and glucose regulation, leading to more consistent and effective blood sugar management for patients with type-2 diabetes.

 

Extended-Release Formulation

 

With its extended half-life, Retatrutide can be administered as a weekly injection, offering patients greater convenience compared to daily medications. This longer duration of action enhances patient compliance and reduces the need for frequent injections, improving the overall treatment experience.

 

High Purity & Stability

 

Retatrutide is synthesized under stringent quality controls, ensuring:

 

● ≥98% purity (by HPLC)

 

● Stable under recommended storage conditions

 

● Free from contaminants such as endotoxins and microbial growth

 

Molecular Details

 

Parameter

Description

CAS Number

2381089-83-2

Molecular Formula

C174H272N50O57S2

Molecular Weight

4057.87 g/mol

Sequence

Not disclosed in full due to intellectual property protections.

Appearance

Lyophilized powder, white to off-white solid

Storage Conditions

Store at -20°C, protected from light

 

Specifications & Packaging

 

Specification

Option

Purity

≥98% (HPLC)

Form

Lyophilized powder

Vial Sizes

1mg, 5mg, 10mg, 50mg vials (bulk or custom packaging options)

Packaging

Individually sealed, sterile packaging with moisture and temperature controls

Shelf Life

24 months from manufacture (when stored at recommended conditions)

 

Applications in Research and Development

 

Retatrutide's mechanism of action makes it an ideal peptide for various metabolic disease research applications, including:

 

● Obesity Research: Understanding the pathways of satiety, fat oxidation, and glucose homeostasis.

 

● Type-2 Diabetes Management: Investigating the dual impact on insulin secretion and glucose control.

 

● Endocrine Regulation: Exploring its combined receptor actions for future therapeutic innovations in diabetes, metabolic disorders, and obesity treatments.

 

● Pharmacokinetic Studies: Examining its long half-life and sustained release profile to improve delivery systems in preclinical models.

 

Retatrutide holds great potential for clinical trials and pharmaceutical development, contributing to drug discovery, early-stage therapeutic formulations, and the optimization of peptide-based treatments.